Farmakologik xususiyatlari
Aminoglikozidlar guruhiga mansub keng ta'sir doirasiga ega antibiotik. Past konsentratsiyalarda bakteriostatik ta'sir ko'rsatadi (30S ribosoma subbirligini bloklaydi va oqsil sintezini buzadi), yuqoriroq konsentratsiyalarda bakterisid ta'sir ko'rsatadi.
Staphylococcusspp. (shu jumladan, Staphylococcusaureus, Staphylococcusepidermidis/koagulaza-manfiy va koagulaza-musbat/ hamda penitsillinga chidamli shtammlar), Streptococcusspp. (shu jumladan, a-b-gemolitik turlar, ayrim negemolitik turlar, Streptococcuspneumoniae); Pseudomonasaeruginosa, Escherichiacoli, Klebsiellapneumoniae, Serratiaspp., Providenciaspp., Shigellaspp., Citrobacterspp., Enterobacteraerogenes, Proteusmirabilis (indol-manfiy) va indol-musbat Proteusspp. turlari, Hemophiliusinfluenzae, Hemophiliusaegyptius, Moraxellalacunata, Acinetobactercalcoaceticus (Herelleavaginacola), ayrim Neisseriaspp. turlari (shu jumladan, Neisseriagonorrhoeae) ga nisbatan yuqori faollikka ega.
Farmakokinetika
Mahalliy qo'llanganda tizimli so'rilishi past.